Eugene Chekler Leaders
Accomplished medicinal chemist and drug hunter: delivered candidates into clinics in Muscular-skeletal and Cardiovascular therapeutic areas. Offer experience with Oncology, Immune-Oncology, Immunology, Kinase Inhibitors design, Epigenetics, Endocrinology, Nuclear Receptors, Gastrointestinal, Protein Misfolding, Antiarrhythmic agents, and unknown mechanism of action. Experience with new therapeutic modalities projects - Protein Degradation (PROTAC), ADCs. Oversee internal lab activities and CROs; external collaborations management experience. Documented success: 42 publications and patent applications; clinical candidate first time disclosure talk.
SELECTED HIGHLIGHTS
Clinical candidate repurposing
Project and Team Leadership
Chemical Biology
Personnel Management
Leading Cross-site Drug Discovery Teams
Structure Based Drug Design
Academic Collaborations
Fragment Based Drug Design
